S-38093
Cat.No:IS2550 Solarbio
CAS:862896-30-8
Molecular Formula:C17H24N2O2
Molecular Weight:288.38
Storage:Powder:2-8℃,2 years;Insolvent(Mother Liquid):-20℃,6 months;-80℃,1 year
Purity:≥98%
Appearance:White to off-white Solid
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S-38093CAS:862896-30-8
Molecular Formula:C17H24N2O2
Molecular Weight:288.38
Storage:Powder:2-8℃,2 years;Insolvent(Mother Liquid):-20℃,6 months;-80℃,1 year
Purity:≥98%
Appearance:White to off-white Solid
Qty:
Size:
CAS | 862896-30-8 |
Name | S-38093 |
Molecular Formula | C17H24N2O2 |
Molecular Weight | 288.38 |
Solubility | Soluble in DMSO(Need ultrasonic) |
Purity | ≥98% |
Appearance | White to off-white Solid |
Storage | Powder:2-8℃,2 years;Insolvent(Mother Liquid):-20℃,6 months;-80℃,1 year |
MDL | MFCD31560487 |
SMILES | C1CC2CN(CC2C1)CCCOC3=CC=C(C=C3)C(=O)N |
InChIKey | MRNMYWNBLVJWKG-UHFFFAOYSA-N |
InChI | InChI=1S/C17H24N2O2/c18-17(20)13-5-7-16(8-6-13)21-10-2-9-19-11-14-3-1-4-15(14)12-19/h5-8,14-15H,1-4,9-12H2,(H2,18,20) |
PubChem CID | 11380684 |
Target Point | Histamine H3 Receptor |
Passage | GPCR & G Protein;Neuronal Signaling;Immunology & Inflammation |
Background | It is an H3 receptor antagonist. |
Biological Activity | S-38093 是一种脑穿透性口服活性 H3 受体拮抗剂,对大鼠、小鼠和人类 H3 受体的 Kis 值分别为 8.8、1.44 和 1.2 μM。[1-2] |
Data Literature Source | [1]. Guilloux JP,et al. S 38093,a histamine H3 antagonist/inverse agonist,promotes hippocampal neurogenesis and improves context discrimination task in aged mice. Sci Rep. 2017 Feb 20;7:42946. [2]. Sors A,et al. Mechanistic characterization of S 38093,a novel inverse agonist at histamine H3 receptors. Eur J Pharmacol. 2017 May 15;803:11-23. |
Unit | Bottle |
Specification | 1mg |
Remark:These protocols are for reference only. Solarbio does not independently validate these methods.
Note:
1. The products are all for scientific research use only. Do not use it for medical, clinical diagnosis or treatment, food and cosmetics, etc. Do not store them in ordinary residential areas.
2. For your safety and health, please wear laboratory clothes, disposable gloves and masks.
3. The experimental results may be affected by many factors, after-sale service is limited to the product itself and does not involve other compensation.
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