Tasimelteon
Cat.No:IT2480 Solarbio
CAS:609799-22-6
Molecular Formula:C15H19NO2
Molecular Weight:245.32
Storage:Powder:2-8℃,2 years;Insolvent(Mother Liquid):-20℃,6 months;-80℃,1 year
Purity:≥98%
Appearance:White to off-white Solid
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TasimelteonCAS:609799-22-6
Molecular Formula:C15H19NO2
Molecular Weight:245.32
Storage:Powder:2-8℃,2 years;Insolvent(Mother Liquid):-20℃,6 months;-80℃,1 year
Purity:≥98%
Appearance:White to off-white Solid
Qty:
Size:
CAS | 609799-22-6 |
Name | Tasimelteon |
Molecular Formula | C15H19NO2 |
Molecular Weight | 245.32 |
Solubility | Soluble in DMSO(Need ultrasonic) |
Purity | ≥98% |
Appearance | White to off-white Solid |
Storage | Powder:2-8℃,2 years;Insolvent(Mother Liquid):-20℃,6 months;-80℃,1 year |
MDL | MFCD09033789 |
SMILES | CCC(=O)NCC1CC1C2=C3CCOC3=CC=C2 |
InChIKey | PTOIAAWZLUQTIO-GXFFZTMASA-N |
InChI | InChI=1S/C15H19NO2/c1-2-15(17)16-9-10-8-13(10)11-4-3-5-14-12(11)6-7-18-14/h3-5,10,13H,2,6-9H2,1H3,(H,16,17)/t10-,13+/m0/s1 |
PubChem CID | 10220503 |
Target Point | Melatonin Receptor |
Passage | GPCR & G Protein;Neuronal Signaling |
Background | It is a selective dual melatonin receptor agonist. |
Biological Activity | Tasimelteon 是一种选择性双重褪黑激素受体激动剂(DMRA),对 MT2 受体的亲和力是 MT1 受体的 2.1-4.4 倍,具有治疗非 24 小时睡眠-觉醒障碍(Non-24)的潜力。[1-2] |
Data Literature Source | [1]. Lavedan C,et al. Tasimelteon: a selective and unique receptor binding profile. Neuropharmacology. 2015 Apr;91:142-7. [2]. Keating GM. Tasimelteon: A Review in Non-24-Hour Sleep-Wake Disorder in Totally Blind Individuals. CNS Drugs. 2016 May;30(5):461-8. |
Unit | Bottle |
Specification | 5mg 10mg |
Remark:These protocols are for reference only. Solarbio does not independently validate these methods.
Note:
1. The products are all for scientific research use only. Do not use it for medical, clinical diagnosis or treatment, food and cosmetics, etc. Do not store them in ordinary residential areas.
2. For your safety and health, please wear laboratory clothes, disposable gloves and masks.
3. The experimental results may be affected by many factors, after-sale service is limited to the product itself and does not involve other compensation.
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