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My Cart> Small Molecule Compounds > Inhibitors & Antagonists & Agonists > Neuronal Signal Pathway > Tiapride HydrochlorideCAS：51012-33-0
Molecular Formula：C15H25ClN2O4S
Molecular Weight：364.89
Storage：Powder:2-8℃，2 years;Insolvent(Mother Liquid):-20℃，6 months;-80℃，1 year
Purity：≥98%
Appearance：White to off-white Solid
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| CAS | 51012-33-0 |
| Name | Tiapride Hydrochloride |
| Molecular Formula | C15H25ClN2O4S |
| Molecular Weight | 364.89 |
| Solubility | Soluble in DMSO(Need ultrasonic) |
| Purity | ≥98% |
| Appearance | White to off-white Solid |
| Storage | Powder:2-8℃，2 years;Insolvent(Mother Liquid):-20℃，6 months;-80℃，1 year |
| EC | EINECS 256-908-4 |
| MDL | MFCD00133861 |
| SMILES | CCN(CC)CCNC(=O)C1=C(C=CC(=C1)S(=O)(=O)C)OC.Cl |
| InChIKey | OTFDPNXIVHBTKW-UHFFFAOYSA-N |
| InChI | InChI=1S/C15H24N2O4S.ClH/c1-5-17(6-2)10-9-16-15(18)13-11-12(22(4，19)20)7-8-14(13)21-3;/h7-8，11H，5-6，9-10H2，1-4H3，(H，16，18);1H |
| PubChem CID | 5702214 |
| Target Point | Dopamine Receptor |
| Passage | Neuronal Signaling;GPCR & G Protein |
| Background | It is a selective D2 and D3 dopamine receptor antagonist with anti-motor dyskinesia and anti-anxiety activities that can be used in the study of neuroleptics. |
| Biological Activity | Tiapride Hydrochloride 是一种选择性口服的 D2 和 D3 多巴胺受体拮抗剂，IC50 值分别为 110-320 nM 和 180 nM，还具有镇静活性和抗焦虑活性。[1-2] |
| IC50 | D2 Receptor: 110-320nM(IC50);D3 Receptor: 180nM(IC50)[1] |
| Data Literature Source | [1]. Scatton B，et al. The preclinical pharmacologic profile of tiapride. Eur Psychiatry. 2001 Jan;16 Suppl 1:29s-34s. [2]. Peters DH，et al. Tiapride. A review of its pharmacology and therapeutic potential in the management of alcohol dependence syndrome. Drugs. 1994 Jun;47(6):1010-32. |
| Unit | Bottle |
| Specification | 50mg 100mg |
Remark：These protocols are for reference only. Solarbio does not independently validate these methods.
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