CAS:1435938-25-2
Storage:Powder:-20℃,2 years;Insolvent(Mother Liquid):-20℃,6 months;-80℃,1 year
Purity:≥98%
Appearance:White to off-white Solid
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JTV-519 hemifumarateCAS:1435938-25-2
Storage:Powder:-20℃,2 years;Insolvent(Mother Liquid):-20℃,6 months;-80℃,1 year
Purity:≥98%
Appearance:White to off-white Solid
CAS | 1435938-25-2 |
English Name | JTV-519 hemifumarate |
Synonyms | K201hemifumarate |
Molecular Formula | C25H32N2O2S·1/2C4H4O4 |
Molecular Weight | 482.64 |
Solubility | Soluble in --- |
Purity | ≥98% |
Appearance | White to off-white Solid |
Storage | Powder:-20℃,2 years;Insolvent(Mother Liquid):-20℃,6 months;-80℃,1 year |
SMILES | COC1=CC2=C(C=C1)SCCN(C2)C(=O)CCN3CCC(CC3)CC4=CC=CC=C4.COC1=CC2=C(C=C1)SCCN(C2)C(=O)CCN3CCC(CC3)CC4=CC=CC=C4.C(=C/C(=O)O)C(=O)O |
InChIKey | MNAIJOCDPCXVEY-WXXKFALUSA-N |
InChI | InChI=1S/2C25H32N2O2S.C4H4O4/c2*1-29-23-7-8-24-22(18-23)19-27(15-16-30-24)25(28)11-14-26-12-9-21(10-13-26)17-20-5-3-2-4-6-20;5-3(6)1-2-4(7)8/h2*2-8,18,21H,9-17,19H2,1H3;1-2H,(H,5,6)(H,7,8)/b;;2-1+ |
PubChem CID | 91885458 |
Target Point | SERCA;ryanodine receptor (RyR) |
Passage | Membrane Transporter&Ion Channel;Neuronal Signaling |
Background | JTV-519 hemifumarate is a Ca2+ dependent blocker of Ca2+ -stimulated ATPase (SERCA) in the sarcoplasmic reticulum. JTV-519 hemifumarate is a partial agonist of the non-self ryanodine receptors in the striated muscle. |
Unit | Bottle |
Specification | 1mg |