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Hypoxia small molecule compound Kit-2

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Hypoxia small molecule compound Kit-2
Cat.No:
IK-HIF-2
Brand:
Solarbio
SKU Tongzhou Beijing Haidian Beijing Wuhan Guangzhou
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CAS号

产品货号

产品名称

分子式

分子量

对应靶点

产品描述

23180-57-6

IP0030

Paeoniflorin;芍药苷

C23H28O11

480.46

HIF/HIF Prolyl-Hydroxylase

据报道,芍药苷可通过mTOR依赖的通路抑制 HIF-1α

89464-63-1

ID0540

DMOG;二甲基乙二酰氨基乙酸

C6H9NO5

175.14

HIF/HIF Prolyl-Hydroxylase

是竞争型的 HIF-1α脯氨酰羟化酶 (HIF-PH) 抑制剂。

5302-45-4

IO0320

β-n-Oxalylamino-l-alanine;三七素

C5H8N2O5

176.13

HIF/HIF Prolyl-Hydroxylase

是一种HIF-prolyl hydroxylase-2 (PHD-2) 抑制剂

808118-40-3

IR0420

Roxadustat;可博美

C19H16N2O5

352.34

HIF/HIF Prolyl-Hydroxylase

Roxadustat 是一种脯氨酰羟化酶 HIF 抑制剂。

38520-57-9

IA4520

N-Acetylcysteine AmideN-乙酰-L-胱氨酸

C5H10N2O2S

162.21

HIF-1α

是一种抗氧化剂,具有消炎活性,能够调节NF-κB的激活、HIF-1αROS

53123-88-9

IR0010

Rapamycin;雷帕霉素

C51H79NO13

914.18

mTOR

是一种有效且特异性的mTOR 抑制剂和自噬激活剂。

38748-32-2

IT0310

Triptolide;雷公藤甲素

C20H24O6

360.4

NF-κB

NF-κB 活化的抑制剂。

284461-73-0

IS0220

Sorafenib;索拉非尼

C21H16ClF3N4O3

464.83

Raf

Raf-1B-Raf的多重激酶抑制剂,还可抑制VEGFR-2VEGFR-3PDGFR-βFlt-3c-KIT

117-39-5

IQ0010

Quercetin;槲皮素

C15H10O7

302.24

PI3K

是一种Sirt1激活剂同时也是PI3K抑制剂

35825-57-1

IC0590

Cryptotanshinone;隐丹参酮

C19H20O3

296.36

STAT

是一种STAT3抑制剂

本套装精选了数种常用于细胞氧感应相关研究的化合物,便于客户进行初筛等操作。客户也可根据自己的需求灵活定制专属Kit。
1. 具有良好的生物活性,且为小包装规格,可用于初筛、预实验、初步验证等操作
2. 靶向HIF/HIF Prolyl-Hydroxylase、mTOR、NF-κB、Raf、PI3K、STAT
3. 可用于探索细胞氧感应相关的研究,例如:缺氧、氧化应激等
4. 客户可根据自己的实验需求灵活定制Kit:规格、套装组成、产品种类、数量、形式(溶液/干粉)均可定制。


Remark:
These protocols are for reference only. Solarbio does not independently validate these methods.

Note:
1. The products are all for scientific research use only. Do not use it for medical, clinical diagnosis or treatment, food and cosmetics, etc. Do not store them in ordinary residential areas.
2. For your safety and health, please wear laboratory clothes, disposable gloves and masks.
3. The experimental results may be affected by many factors, after-sale service is limited to the product itself and does not involve other compensation.
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