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ER STRESS small molecule compound Kit-1

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ER STRESS small molecule compound Kit-1
Cat.No:
IK-ERS-1
Brand:
Solarbio
SKU Tongzhou Beijing Haidian Beijing Wuhan Guangzhou
IK-ERS-1-10*1ml Inquiry Inquiry Inquiry Inquiry
IK-ERS-1-10*2mg Inquiry Inquiry Inquiry Inquiry
IK-ERS-1-10*5mg Inquiry Inquiry Inquiry Inquiry
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CAS号

产品货号

产品名称

分子式

分子量

对应靶点

产品描述

27208-80-6

IP0770

Polydatin;虎杖苷

C20H22O8

390.38

ER Stress

存在于传统中药虎杖根中,在多个实验模型中具有抗炎作用。据报道,可抑制G6PD,并诱导氧化和内质网应激

14605-22-2

IT0790

Tauroursodeoxycholic acid;牛磺熊去氧胆酸

C26H45NO6S

499.7

ER Stress

是一种内质网应激抑制剂。

35807-85-3

IT0370

Tauroursodeoxycholate Sodium;牛磺熊去氧胆酸钠

C26H44NNaO6S

521.69

ER StressCaspase

是一种内质网应激抑制剂,可显著降低凋亡分子如 caspase-3 caspase-12 表达。

1716-12-7

IS0080

Sodium 4-phenylbutyrate4-苯基丁酸钠盐

C10H11NaO2

186.18

ER Stress

是一种组蛋白去乙酰化酶 (HDAC) 和内质网应激 (ER) 抑制剂,可用于癌症和感染等疾病的研究。

73-31-4

IM0080

Melatonin;褪黑素

C13H16N2O2

232.28

ATF6

是一种激素,可激活褪黑激素受体。也是一种新型的选择性 ATF-6 抑制剂。

1589527-65-0

IK0470

KIRA6

C28H25F3N6O

518.53

IRE1

是有效的IIIRE1α激酶抑制剂。

14003-96-4

IM2400

8-Formyl-7-Hydroxy-4-Methyl-Coumarin8-甲酰基-7-羟基-4-甲基香豆素

C11H8O4

204.18

IRE1

是高效的选择性IRE1 Rnase抑制剂。

307543-71-1

IS1990

STF083010

C15H11NO3S2

317.38

IRE1

是一种特异性IRE1α endonuclease抑制剂。

1337532-29-2

IG1320

GSK2656157

C23H21FN6O

416.45

PERK

是选择性,ATP竞争性的 PERK 抑制剂。

1337531-36-8

IG1330

GSK2606414

C24H20F3N5O

451.44

PERK

PERK 抑制剂。

本套装精选了数种常用于内质网应激相关研究的化合物,便于客户进行初筛等操作。客户也可根据自己的需求灵活定制专属Kit。
1. 具有良好的生物活性,且为小包装规格,可用于初筛、预实验、初步验证等操作
2. 靶向ER Stress、ATF6、IRE1、PERK
3. 可用于探索内质网应激的相关研究
4. 客户可根据自己的实验需求灵活定制Kit:规格、套装组成、产品种类、数量、形式(溶液/干粉)均可定制。


Remark:
These protocols are for reference only. Solarbio does not independently validate these methods.

Note:
1. The products are all for scientific research use only. Do not use it for medical, clinical diagnosis or treatment, food and cosmetics, etc. Do not store them in ordinary residential areas.
2. For your safety and health, please wear laboratory clothes, disposable gloves and masks.
3. The experimental results may be affected by many factors, after-sale service is limited to the product itself and does not involve other compensation.
SERVICE FOR SCIENTIFIC RESEARCH,RESPONSIBLE FOR LIFE
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